Aromatase Inhibitors for Men: Buy Estrogen Blockers Online
Aromatase Inhibitors first inhibit the enzyme aromatase, which is responsible for converting testosterone to estrogen; second, they dock onto estrogen receptors, preventing stronger forms of estrogen from docking. Estrogen blockers are thus divided into aromatase inhibitors and estrogen receptor blockers.
Aromatase inhibitors are also called estrogen blockers or estrogen inhibitors. So both are the same thing, only the name is different.
Aromatase inhibitors and estrogen blockers for gynecomastia
Not pretty, but unfortunately a reality for some men. Gynecomastia, or female breasts, is caused by fat accumulation on the breasts, the appearance reminds more of soft female breasts than hard man muscles. However, estrogen blockers can also be quite helpful in reducing the fat on the breasts and solving the problem with gynecomastia.
How to use them
- Arimidex (chemical name anastrozole)
- Aromazine (chemical name exemestane)
- Alvogen (chemical name letrozole)
The simplest method: each tablet is taken once a day. All three are available as generic medicines. Aromatase blockers can be given to men with breast cancer or gynecomastia, although another medicine called tamoxifen is often used.
What are aromatase inhibitors or blockers?
Aromatase inhibitors are a class of medicines that lower levels of estrogen (female sex hormones) in the blood and increase levels of testosterone and gonadotropic hormones. These medicines are often used to treat and prevent the development of gynecomastia in men.
The medicines are commonly used in elite sports, where estrogenic effects are often associated with the use of anabolic steroids. They are taken to:
- Reduce the risk of gynecomastia;
- Increase the concentration of anabolic hormones in the body;
- Creating an attractive muscle relief, which is achieved by reducing the negative effects of estrogen;
- Prevention of hypertension;
- Reducing the influence of estrogen on the hypothalamic-pituitary-testicular axis, speeding up the body's recovery.
When composing a cycle, it should be taken into account that not all anabolic steroids are aromatase. Treatment with aromatase blockers is useful if an athlete takes testosterone derivatives, methandienone, methyltestosterone.
Boldenone and Halotestin are slightly aromatized.
Some of the most affordable and popular products in this category are:
- Letrozole
- Arimidex (Anastrozole)
- Exemestane (Aromasin)
- Tamoxifen
- Proviron
At the same time, it should be emphasized that a moderate level of estrogen in the blood has a positive effect on the athlete's body and promotes the growth of muscle mass. Therefore, prophylactic dosages are indicated in quantities that allow maintaining normal physiological hormone levels in members of the stronger sex.
How athletes use it
Most athletes begin taking aromatase inhibitors for men only when the first symptoms of gynecomastia appear. The pathology manifests itself in the form of swelling, itching in the area of the nipples, redness of the breasts. However, this option of using medicine can not be considered correct and optimal.
A much better solution would be to visit a medical facility and get tested for estradiol levels 10 days after starting a steroid regimen with anabolic steroids, which have a short half-life. If the athlete has chosen to inject longer esters, the test is done 3-4 weeks later. After receiving the results, the specialist may prescribe 0.5 mg of anastrozole every 2 days. After 10 days, a control test is performed, the results of which allow the specialist to adjust the dose.
Another way to use aromatase blockers is to take moderate or low doses, taking into account the individual sensations of the athlete. If the bodybuilder notices a decrease in libido, erection problems or depressive states after starting the course, the dose is reduced.
Side effects
The side effects of aromatase inhibitors can occur in a number of cases. For example, a moderate concentration of estrogen concentration in the blood is also good for the male body. Steroids containing female sex hormones have a positive effect on the sensitivity of androgen receptors, which increases the effectiveness of anabolic steroids.
Practice shows that excessive fascination with blockers can lead to a sharp drop in estrogen levels, so it is important to know and understand how to take aromatase inhibitors. Neglecting medical advice can lead to a sharp drop:
- Slowing and complete cessation of muscle growth;
- Development of arthralgia, which manifests itself mainly in joint pain;
- Decrease in the strength of bone tissue, increase in the risk of injury;
- Increase in "bad" cholesterol;
- Deterioration of the quality of sexual life;
- Destabilization of the psycho-emotional state, mood swings and depression.
It is important to take aromatase blockers in tablet form under constant supervision of qualified professionals.
Pharmacological information
Anastrozole is one of the most popular medicines in this category. The price of the aromatase inhibitor of this category is fully justified by its positive properties. The substance is one of the strong, highly selective non-steroidal medicines recommended for both athletes and post-menopausal women to reduce the amount of estradiol.
Depending on the manufacturer, the medicine is produced in packs of 14, 20, 28, or 50 tablets of 1 mg. It is taken orally 1 mg once a day. The active substances are quickly absorbed through the gastrointestinal tract, and the maximum concentration in the blood is detected within 2 hours after taking on an empty stomach. It is recommended to take the medicine in the morning, as simultaneous intake of food slightly reduces the beneficial properties and slows down its absorption. The elimination half-life is 40-50 hours, and about 10% of the dose is excreted from the body naturally unchanged.
Adverse effects of intake include dry mucous membranes in the genitourinary area, flushing, deterioration of hair quality, liver dysfunction, appearance of skin problems. Anorexia, nausea, vomiting or diarrhea may occur. At the same time, the negative effects of taking it occur quite rarely. To avoid this, it is enough to buy good quality aromatase inhibitors and take them according to the instructions. In bodybuilding, this substance is used to reduce the risk of gynecomastia and prevent excessive fluid accumulation in the tissues.
Letrozole is another competitive inhibitor. Compared to the previous medicine, it decreases estrogen concentration more (up to 98.8%). As a rule, experts recommend oral intake of 1 tablet per day, regardless of meals.
The active substances are rapidly absorbed in the gastrointestinal tract. Equilibrium concentration occurs 4 weeks after the start of treatment. About 60% of the medicine binds to plasma proteins, and in erythrocytes the concentration reaches 80%. It is excreted naturally in the urine. The medicine is strictly contraindicated in liver problems.
Most side effects are mild, most of the list is similar to anastrozole. In addition, a small number of women may begin to have bloody vaginal discharge, leucorrhea, and increased levels of sweating and shortness of breath.
Exemestane, which reduces estrogen production by 97%, belongs to the third generation of inhibitors
How to buy aromatase inhibitors online?
The advantage of buying estrogen blockers online in our store is the fact that the price is the cheapest you can find, and you can buy directly without a prescription. We are the number one in sports pharmacology and we do everything to make our customers appreciate us.
If you have not decided exactly which supplements to buy for your workout, you can contact our consultants. We will help you determine the preparation you need from the range of aromatase inhibitors. Exact course of taking such medicines should still be determined by your personal trainer.
